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Updated: Jun 13, 2026

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Skeletal Editing of 4-Substituted Isothiazoles to Pyrazoles Via a Two-Atom N-S to N-N Swap

Bao-Qin Huang1, Jin-Zhen Xu1, Zi-Cheng Huang1

  • 1State Key Laboratory of Anti-Infective Drug Discovery and Development; Guangdong Provincial Key Laboratory of Chiral Molecules and Drug Discovery, School of Pharmaceutical Sciences, Sun Yat-sen University; Guangzhou, 510006, China.

Organic Letters
|June 12, 2026
PubMed

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