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High-Throughput Cellular Profiling of Targeted Protein Degradation Compounds Using HiBiT CRISPR Cell Lines
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On-Demand Activatable PROTACs for Targeted Protein Degradation

Caiyun Guo1, Zhibin Ren1, Xiaomei Wu1

  • 1State Key Laboratory of Chemical Resource Engineering, MOE Key Lab of Biomedical Materials of Natural Macromolecules, Beijing University of Chemical Technology, Beijing, China.

Chemistry (Weinheim an Der Bergstrasse, Germany)
|June 20, 2026
PubMed
Abstract

Keywords:
PROTACsactivationcancerprodrugtargeted protein degradation

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