C3-H methylenephosphonylation of azaarenes enabled by catalyst-controlled regioselective cyclizative rearrangement

Dan Liu1, Fang-Zhou Li1, Yu-Ping He2

  • 1Shanghai Key Laboratory for Molecular Engineering of Chiral Drugs, Shanghai Frontiers Science Center for Drug Target Identification and Delivery, and Laboratory of Innovative Immunotherapy, School of Pharmaceutical Sciences, Shanghai Jiao Tong University Shanghai 200240 China hua.wu@sjtu.edu.cn.

Chemical Science
|June 22, 2026
PubMed

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