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Updated: Jun 28, 2026

High-Throughput Cellular Profiling of Targeted Protein Degradation Compounds Using HiBiT CRISPR Cell Lines
05:33

High-Throughput Cellular Profiling of Targeted Protein Degradation Compounds Using HiBiT CRISPR Cell Lines

Published on: November 9, 2020

Development of APH003─a Highly Potent, Selective, and Orally Bioavailable IRAK4 PROTAC Degrader for the Treatment of

Xi-Wei Wu1,2, Zhao-Min Chen2, Cui Gao2

  • 1School of Pharmaceutical Sciences, Sun Yat-Sen University, Guangzhou 510006, China.

Journal of Medicinal Chemistry
|June 26, 2026
PubMed

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