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Covalent Fragment Screening Using the Quantitative Irreversible Tethering Assay
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Stereoselective Covalent Targeting of BTK(C481S) and Kinases with β-Lactone Electrophiles

Celine D Wang1,2, Polina E Barzova1, Julian Robles1

  • 1Department of Chemistry, University of California, Berkeley, California 94720, USA.

Biorxiv : the Preprint Server for Biology
|July 17, 2026
PubMed
Abstract

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