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A Direct, Early Stage Guanidinylation Protocol for the Synthesis of Complex Aminoguanidine-containing Natural Products
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Conversion of artemisinin into novel unprotected N-alkylamine-11-azaartemisinins with enhanced antimalarial activity

Komal Rathi1, Aashima Gupta2, Priyanka Yadav1

  • 1Department of Chemistry, Banasthali University, Banasthali Newai 304022, Rajasthan, India.

Bioorganic & Medicinal Chemistry Letters
|July 22, 2026
PubMed

Keywords:
AntimalarialArtemisininAzaartemisininPlasmodium falciparum

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