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Updated: Aug 5, 2026

Real-time Imaging of Leukotriene B4 Mediated Cell Migration and BLT1 Interactions with β-arrestin
13:45

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Published on: December 23, 2010

A Structure-guided Active Site Affinity Ligand Unmasks a Stress-Sensitizing Role for BLVRB in the Endoplasmic

Rahul Raghavan Thekke Veedu1,2, Jawaad Sheriff1, Natasha M Nesbitt1

  • 1Blood Cell Technologies, JLABS@NYC, 101 Sixth Avenue, New York, New York 10013, United States.

Journal of Medicinal Chemistry
|July 27, 2026
PubMed
Summary

Biliverdin IXb reductase (BLVRB) activity was measured in real-time using a novel nanoBRET platform. This technology allows for precise analysis of BLVRB inhibitors and their role in cellular stress responses.

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