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Updated: Aug 5, 2026

Protocol for the Synthesis of Ortho-trifluoromethoxylated Aniline Derivatives
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Click Chemistry Approach to Derivatisation of Fluconazole

Michał Janowski1, Oleg M Demchuk2, Sylwia Andrzejczuk3

  • 1Doctoral School, Medical University of Lublin, Chodzki 7, 20-093 Lublin, Poland.

Molecules (Basel, Switzerland)
|July 28, 2026
PubMed

Keywords:
1,2,3-triazoles1,2,4-triazolesCuAACantifungal agentsazide-alkyne Huisgen cycloadditionclick chemistrycopper catalysisdrug modificationfluconazole

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