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Intensification versus combination: revisiting the past and envisioning the future of LDHA inhibitors

Weixi Yuan1, Qiang Kang2, Yin Zhao1

  • 1The First Affiliated Hospital, Department of Pharmacy, Institute of Pharmacy and Pharmacology, Hengyang Medical School, University of South China, Hengyang, 421001, Hunan, China.

Cancer Chemotherapy and Pharmacology
|August 20, 2026
PubMed

Keywords:
Cancer therapeuticsChemoresistanceDrug combination strategyLDHA inhibitorsLactate dehydrogenase AMetabolic reprogrammingTumor metabolismWarburg effect

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