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Updated: Aug 22, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
07:41

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Pharmacological targeting of GCN5/PCAF (KAT2A/B): current drug discovery strategies and translational potential

Priyanka Pandey1, Prajjval Mishra1, Pritam Biswas2

  • 1Transcription and Disease Laboratory, Molecular Biology and Genetics Unit, Jawaharlal Nehru Centre for Advanced Scientific Research, Jakkur, Bengaluru 560064, India.

Drug Discovery Today
|August 20, 2026
PubMed

Keywords:
GCN5/PCAFGNAT familyepigenetic regulationlysine acetyltransferasestherapeutic implications

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