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Updated: Sep 3, 2026

A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones
07:30

A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones

Published on: January 21, 2020

Strategic Use of the Necessary Nitrogen Atom for Holistic Property-Based Drug Design

Lewis D Pennington1, Julia M Clay1, Sandrine M Hell1

  • 1Drug Hunter , Portland, Oregon97204, United States.

Journal of Medicinal Chemistry
|September 1, 2026
PubMed

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