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Technical Aspect of the Automated Synthesis and Real-Time Kinetic Evaluation of [11C]SNAP-7941
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First-in-Human Phase I Trial of HRS-2129, a Selective Nav1.8 Inhibitor: Safety, Tolerability, Pharmacokinetics, and

Jie Huang1,2,3,4, Qian Wu2,3, Saiying Wang5

  • 1Xiangya School of Pharmaceutical Sciences, Central South University, Changsha, Hunan, People's Republic of China.

Drug Design, Development and Therapy
|September 9, 2026
PubMed
Abstract

Keywords:
HRS-2129Nav1.8 inhibitorhealthy subjectspain tolerancepharmacokineticsphase I clinical trialsafety

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