Related Experiment Video

Updated: Oct 16, 2026

A Semi-High-Throughput Adaptation of the NADH-Coupled ATPase Assay for Screening Small Molecule Inhibitors
10:28

A Semi-High-Throughput Adaptation of the NADH-Coupled ATPase Assay for Screening Small Molecule Inhibitors

Published on: August 17, 2019

Research progress on ATP-citrate lyase and its inhibitors: a metabolic-epigenetic perspective

Qinglin Liu1, Hongbin Sun1,2, Liang Dai1,2

  • 1Jiangsu Key Laboratory of Drug Discovery for Metabolic Disease, State Key Laboratory of Natural Medicines, China Pharmaceutical University, Nanjing, China.

Journal of Enzyme Inhibition and Medicinal Chemistry
|October 14, 2026
PubMed

Keywords:
ACLY inhibitorsATP-citrate lyasedrug discoverystructural biologystructure-activity relationships

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