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Targeting Transcriptional Coactivators p300/CBP: Small-Molecule Inhibitors or Bifunctional Proximity-Inducing

Zonglong Chen1, Xun Huang2,3,4,5, Yingxia Li1

  • 1Department of Medicinal Chemistry, School of Pharmacy, Fudan University, 826 Zhangheng Road, Shanghai201203, China.

Journal of Medicinal Chemistry
|October 23, 2026
PubMed

Keywords:
bifunctional proximity-inducing modalitybromodomainhistone acetyltransferasep300/CBPsmall-molecule inhibitortranscriptional coactivator

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