Related Experiment Video

Updated: Oct 25, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
07:41

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

Published on: February 20, 2018

Development of Potent G Protein Pathway-Biased GPR183 Agonists

Kaustubh R Bhuskute1, Asmita Manandhar1, Viktoria M S Kjær2

  • 1Department of Drug Design and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Jagtvej 162, 2100Copenhagen, Denmark.

Journal of Medicinal Chemistry
|October 23, 2026
PubMed

Keywords:
7α,25-OHCEBI2G proteinGPR183TUG-2604biased agonistsbiased signalingdendritic cell migrationoxysterolreceptorβ-arrestin

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