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System for Efficacy and Cytotoxicity Screening of Inhibitors Targeting Intracellular Mycobacterium tuberculosis
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Antivirulence Benzothiophenes Inhibit Intracellular Mycobacterium tuberculosis by Targeting the Sensor Histidine

Vladislav Lobanov1, Andréanne Lupien2, Anthony Vocat2

  • 1Research Centre of Biotechnology RAS , 33-2 Leninsky Prospect, 119071Moscow, Russia.

Journal of Medicinal Chemistry
|October 23, 2026
PubMed

Keywords:
ESX-1 systemanti-infective agentbenzothiophenehistidine kinase MprBmycobacterial virulencepathoblockertuberculosisvirulence inhibitor

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