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Updated: Oct 28, 2026

Characterizing Modulators of Protease-Activated Receptors with a Calcium Mobilization Assay Using a Plate Reader
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Characterizing Modulators of Protease-Activated Receptors with a Calcium Mobilization Assay Using a Plate Reader

Published on: May 24, 2024

Store-Operated Calcium Entry Inhibitors: Structural Diversity, Mechanisms of Action, and Optimization Strategies

Anastasiia A Zakharova1, Dmitriy A Grekhnev1, Elena V Kaznacheyeva1,2

  • 1Institute of Cytology of Russian Academy of Science, Tikhoretsky Ave. 4, 194064 St. Petersburg, Russia.

International Journal of Molecular Sciences
|October 27, 2026
PubMed

Keywords:
OraiSOC channel inhibitorsSOCESTIMcalciumstore-operated calcium entrystructure–activity relationship

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