Natural dehydrocostus lactone-based analogues as new structural PDPK1 allosteric activators against HBV

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Identifying Inhibitors of the HBx-DDB1 Interaction Using a Split Luciferase Assay System
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Identifying Inhibitors of the HBx-DDB1 Interaction Using a Split Luciferase Assay System

Published on: December 21, 2019

Hang Sun1, Yu-Jing Mao1, Dan-Yang Zhu1

  • 1Yunnan Key Laboratory of Cross-Border Infectious Disease Control and Prevention and Novel Drug Development (Under Construction), Center for Pharmaceutical Sciences, Faculty of Life Science and Technology, Kunming University of Science and Technology, Chenggong Campus, Kunming, 650500, China.

European Journal of Medicinal Chemistry
|November 4, 2026
PubMed

Keywords:
Dehydrocostus lactoneHBVOptimizationPDPK1Sesquiterpene derivative

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