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Precision of digoxin radioimmunoassays and matrix effects: four kits compared

Clinical Biochemistry
|April 1, 1981
PubMed

Insights

Sample matrix interference affects digoxin radioimmunoassays. Different patient conditions, like spironolactone use or uremia, caused significant digoxin measurement errors, impacting clinical accuracy.

Area of Science:

  • Clinical Chemistry
  • Analytical Chemistry
  • Pharmacokinetics

Background:

  • Accurate digoxin measurement is crucial for therapeutic drug monitoring.
  • Radioimmunoassays are commonly used for digoxin quantification.
  • Potential interference from patient sample matrices can affect assay accuracy.

Purpose of the Study:

  • To investigate the impact of sample matrix interference on digoxin radioimmunoassays.
  • To evaluate the performance of four commercial digoxin immunoassay kits.
  • To assess digoxin measurement accuracy in plasma from patients with specific conditions.

Main Methods:

  • Four commercial digoxin radioimmunoassay kits were used.
  • Plasma samples from non-digitalized patients with essential hypertension (on spironolactone), uremia, and acute myocardial infarction (AMI) were analyzed.
  • A known concentration of digoxin (2.50 nmol/L) was added to all samples for interference assessment.

Main Results:

  • Two kits overestimated digoxin in spironolactone-treated patients (p<0.01).
  • One kit underestimated digoxin in uremic patients (p<0.01).
  • One kit overestimated digoxin in AMI patients (p<0.05).
  • Significant inter-assay and intra-assay variations were observed.

Conclusions:

  • Sample matrix significantly interferes with digoxin radioimmunoassays, leading to inaccurate measurements.
  • Assay performance varied considerably between different commercial kits and patient sample types.
  • Despite matrix effects, the overall low precision of the assays made these deviations secondary.

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