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Anipamil prevents ST depression in patients with stable angina pectoris

C T Larsen1, C Sørum, V Rasmussen

  • 1Department of Cardiology, Hvidovre University Hospital, Copenhagen, Denmark.

Insights

Once-daily anipamil effectively treats stable angina by significantly reducing myocardial ischemia. This anti-ischemic drug demonstrates 24-hour efficacy, making it a valuable option for patients with transient myocardial ischemia.

Area of Science:

  • Cardiology
  • Pharmacology

Background:

  • Stable angina pectoris is a common condition characterized by chest pain due to myocardial ischemia.
  • Current treatments aim to reduce the frequency and severity of ischemic episodes.

Purpose of the Study:

  • To evaluate the 24-hour anti-ischemic efficacy of once-daily anipamil in patients with stable angina.
  • To compare the effects of anipamil 80 mg and 160 mg against placebo.

Main Methods:

  • Double-blind, placebo-controlled crossover study design.
  • Inclusion of 19 patients with stable angina and documented ischemia.
  • 24-hour ambulatory ECG monitoring to assess transient myocardial ischemia duration.

Main Results:

  • Anipamil significantly reduced the total duration of transient myocardial ischemia.
  • Anipamil 80 mg reduced ischemia duration to 712 minutes (p < 0.001), with 87% asymptomatic episodes.
  • Anipamil 160 mg reduced ischemia duration to 913 minutes (p > 0.001), with 92% asymptomatic episodes.

Conclusions:

  • Once-daily anipamil is an effective 24-hour anti-ischemic treatment for stable angina.
  • Anipamil demonstrates significant efficacy in reducing both symptomatic and asymptomatic transient myocardial ischemia.

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