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In vitro sensitivity of medically significant Fusarium species to various antimycotics

A S Sekhon1, A A Padhye, A K Garg

  • 1National Centre for Human Mycotic Diseases, University of Alberta Hospitals, Edmonton, Canada.

Chemotherapy
|July 1, 1994
PubMed

Insights

This study evaluated antifungal susceptibility in Fusarium species. Most Fusarium isolates showed susceptibility to amphotericin B and itraconazole, but resistance to fluconazole.

Area of Science:

  • Mycology
  • Antimicrobial Susceptibility Testing

Background:

  • Fusarium species are opportunistic fungal pathogens.
  • Antifungal resistance is a growing concern in managing Fusarium infections.

Purpose of the Study:

  • To determine the in vitro antifungal susceptibility profiles of various Fusarium species.
  • To compare the efficacy of different antifungal agents against Fusarium isolates.

Main Methods:

  • Sixteen Fusarium isolates (F. chlamydosporum, F. equiseti, F. moniliforme, F. oxysporum, F. proliferatum, F. solani) were tested.
  • Antifungal susceptibility was assessed using minimal inhibitory concentration (MIC) and minimal fungicidal concentration (MFC) assays.
  • Tested antifungals included amphotericin B, 5-fluorocytosine, fluconazole, itraconazole, ketoconazole, JAI-amphotericin B, hamycin, and combination therapies.

Main Results:

  • All Fusarium isolates exhibited resistance to 5-fluorocytosine and fluconazole (MIC > 100 µg/ml).
  • Hamycin showed variable efficacy (MIC 12.5-100 µg/ml), with F. equiseti being more susceptible.
  • Amphotericin B, itraconazole, and ketoconazole demonstrated broad activity (MICs ranging from 0.78 to 100 µg/ml).
  • Certain isolates (F. solani, F. oxysporum, F. chlamydosporum, F. equiseti, F. moliniforme) were more susceptible to amphotericin B, itraconazole, ketoconazole, hamycin, and amphotericin B with 5-fluorocytosine.

Conclusions:

  • Fusarium species display significant resistance to fluconazole and 5-fluorocytosine.
  • Amphotericin B and itraconazole are promising agents for treating Fusarium infections.
  • Further research into combination therapies may enhance treatment efficacy.

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