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Structure-activity correlations in a homologous series of 2-substituted isonicotinic acid hydrazides

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Preliminary evaluation of the toxicity and efficacy of novel 2,4-diamino-5-benzylpyrimidine-sulphone derivatives using rat and human tissues in vitro.

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Partial resistance of E. coli mutants against 2, 4-diamino-5-benzylpyrimidines by interactions with bacterial membrane lipopolysaccharides. Derivation of quantitative structure-binding relationships.

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Structure-activity correlations in a homologous series of 2-substituted isonicotinic acid hydrazides

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