Potent thrombin inhibitors that probe the S1 subsite: tripeptide transition state analogues based on a heterocycle-activated carbonyl group

Precision Studies and Searches for CP Asymmetries in the Inclusive Decay Λ_{c}^{+}→ΛX.

Physical review letters·2026

First Energy-Scan Measurement of e^{+}e^{-}→K^{+}K^{-} around the ψ(2S) Resonance.

Physical review letters·2026

Measurements of the Absolute Branching Fraction of the Semileptonic Decay Ξ^{-}→Λe^{-}ν[over ¯]_{e} and the Axial Charge of Ξ^{-}.

Physical review letters·2026

First Experimental Constraint on the Scalar Current in the D^{0(+)}→K[over ¯]ℓ^{+}ν_{ℓ} Transition.

Physical review letters·2026

First Observation of D^{0(+)}→K[over ¯]ωe^{+}ν_{e} and Determination of the Branching Fraction of K[over ¯]_{1}(1270)→K[over ¯]ω.

Physical review letters·2026

Measurement of the Λ electric dipole moment with an entangled baryon-antibaryon system.

Science (New York, N.Y.)·2026

Structural and Mechanistic Studies of ADEPs Yield Potent Antibacterials and a Drug Formulation Strategy for Tuberculosis.

Journal of medicinal chemistry·2026

A 177Lu-Labeled Circular Bivalent Aptamer for PTK7-Targeting Radionuclide Therapy in Ovarian Cancer and Orthotopic Hepatoblastoma.

Journal of medicinal chemistry·2026

From Fragment Hit to Clinical Candidate: Discovery of Dual H1R/H4R Ligands with Superior Efficacy in Allergic Conjunctivitis.

Journal of medicinal chemistry·2026

Potent Anticancer Tethered Organorhodium(III) Complexes Target the Mitochondria.

Journal of medicinal chemistry·2026

Discovery of a Covalent NLRP3 LRR-Domain Probe: Reversing Renal Fibrosis via Immunometabolic Reprogramming in Organoid and Murine Models.

Journal of medicinal chemistry·2026

Lead Optimization of Multimutant KRAS Switch-II Pocket Macrocyclic Inhibitors via Isosteric Replacement to Improve ADME and Oral Exposure.

Journal of medicinal chemistry·2026

Multicomponent synthesis of 2-amino-tetrahydro-4H-chromenes catalyzed by chitosan and evaluation of anti-Leishmania activity.

Future medicinal chemistry·2026

Catalytic Asymmetric Synthesis of Spiro[3.3]heptane-Based Axially Chiral α-Amino Acids.

Angewandte Chemie (International ed. in English)·2026

Phytochemical Profiling, In Vitro α-Amylase Inhibitory and Antioxidant Activities of Madhuca longifolia Leaf and Bark Extracts with Molecular Docking Analysis.

Plants (Basel, Switzerland)·2026

Combined Fungal Elicitor and Methyl Jasmonate Enhance Alkaloid Accumulation in Catharanthus roseus Suspension Cultures: An Integrated Molecular and Phytochemical Study.

Plants (Basel, Switzerland)·2026

The Therapeutic Potential of Berry-Derived and Berry-Based Interventions in Inflammatory Bowel Disease: A Comprehensive Systematic Review of Preclinical and Clinical Evidence.

Nutrients·2026

Integrated Transcriptomic and Network Analysis Identifies Candidate Kinase-Mediated Thyroid-Associated Targets of Withaferin A.

International journal of molecular sciences·2026

Related Experiment Videos

Potent thrombin inhibitors that probe the S1 subsite: tripeptide transition state analogues based on a

Related Concept Videos

Precision Studies and Searches for CP Asymmetries in the Inclusive Decay Λ_{c}^{+}→ΛX.

First Energy-Scan Measurement of e^{+}e^{-}→K^{+}K^{-} around the ψ(2S) Resonance.

Measurements of the Absolute Branching Fraction of the Semileptonic Decay Ξ^{-}→Λe^{-}ν[over ¯]_{e} and the Axial Charge of Ξ^{-}.

First Experimental Constraint on the Scalar Current in the D^{0(+)}→K[over ¯]ℓ^{+}ν_{ℓ} Transition.

First Observation of D^{0(+)}→K[over ¯]ωe^{+}ν_{e} and Determination of the Branching Fraction of K[over ¯]_{1}(1270)→K[over ¯]ω.

Measurement of the Λ electric dipole moment with an entangled baryon-antibaryon system.

Structural and Mechanistic Studies of ADEPs Yield Potent Antibacterials and a Drug Formulation Strategy for Tuberculosis.

A 177Lu-Labeled Circular Bivalent Aptamer for PTK7-Targeting Radionuclide Therapy in Ovarian Cancer and Orthotopic Hepatoblastoma.

From Fragment Hit to Clinical Candidate: Discovery of Dual H1R/H4R Ligands with Superior Efficacy in Allergic Conjunctivitis.

Potent Anticancer Tethered Organorhodium(III) Complexes Target the Mitochondria.

Discovery of a Covalent NLRP3 LRR-Domain Probe: Reversing Renal Fibrosis via Immunometabolic Reprogramming in Organoid and Murine Models.

Lead Optimization of Multimutant KRAS Switch-II Pocket Macrocyclic Inhibitors via Isosteric Replacement to Improve ADME and Oral Exposure.

Multicomponent synthesis of 2-amino-tetrahydro-4H-chromenes catalyzed by chitosan and evaluation of anti-Leishmania activity.

Catalytic Asymmetric Synthesis of Spiro[3.3]heptane-Based Axially Chiral α-Amino Acids.

Phytochemical Profiling, In Vitro α-Amylase Inhibitory and Antioxidant Activities of Madhuca longifolia Leaf and Bark Extracts with Molecular Docking Analysis.

Combined Fungal Elicitor and Methyl Jasmonate Enhance Alkaloid Accumulation in Catharanthus roseus Suspension Cultures: An Integrated Molecular and Phytochemical Study.

The Therapeutic Potential of Berry-Derived and Berry-Based Interventions in Inflammatory Bowel Disease: A Comprehensive Systematic Review of Preclinical and Clinical Evidence.

Integrated Transcriptomic and Network Analysis Identifies Candidate Kinase-Mediated Thyroid-Associated Targets of Withaferin A.

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Potent thrombin inhibitors that probe the S1 subsite: tripeptide transition state analogues based on a...

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Potent thrombin inhibitors that probe the S1 subsite: tripeptide transition state analogues based on a