Lead development: validation and application of high throughput screening for determination of pharmacokinetic parameters for enzyme inhibitors

Induction of spermatogenesis by androgens in gonadotropin-deficient (hpg) mice.

Endocrinology·1995

Dysfibrinogenemia: a case with thrombosis (fibrinogen Richfield) and an overview of the clinical and laboratory spectrum.

American journal of hematology·1995

Purification and properties of four monocot lectins from the family Araceae.

Phytochemistry·1995

Concurrent evaluation of immunization programme by Lot Quality Assurance Sampling.

Journal of tropical pediatrics·1995

Characterization of a low-temperature-induced cDNA from winter Brassica napus encoding the 70 kDa subunit of tonoplast ATPase.

Plant molecular biology·1995

Structural studies on the PH domains of Db1, Sos1, IRS-1, and beta ARK1 and their differential binding to G beta gamma subunits.

Biochemistry·1995

Synthesis of axially chiral benzochalcogenophene derivatives and their anti-proliferative activities in cancer cells.

Bioorganic & medicinal chemistry·2026

Hypoxia-activated 2-nitroimidazole-brusatol carbonate prodrugs for enhanced gastric cancer therapy with reduced systemic toxicity.

Bioorganic & medicinal chemistry·2026

Rivastigmine-centered molecular hybridization strategies for multi-targeted intervention in Alzheimer's disease: Advances (2020-2026).

Bioorganic & medicinal chemistry·2026

Criteria-guided selection of alternative zinc-binding groups of HDAC3 inhibitors using in silico and in vitro approaches.

Bioorganic & medicinal chemistry·2026

Design, synthesis, and biological evaluation of novel dihydropyrimidinone imines as potent anticancer agents targeting AKT to induce cell cycle arrest and apoptosis in breast Cancer cells.

Bioorganic & medicinal chemistry·2026

Design, synthesis, biological and computational evaluation of Thieno[3,2-d]pyrimidine-based inhibitors of JAK3 kinase.

Bioorganic & medicinal chemistry·2026

Quantification of PDGF-AB and TGF-β1 Proteins in Platelet-rich Plasma Obtained under Different Conditions.

Prague medical report·2026

A Multiparametric in vitro Strategy for Small Molecule Drug-Induced Liver Injury Risk Mitigation in Early Drug Development.

Toxicological sciences : an official journal of the Society of Toxicology·2026

A Phase 3, Multicenter, Randomized, Placebo-Controlled Trial Evaluating the Efficacy, Safety, and Tolerability of Serdexmethylphenidate/d-Methylphenidate Capsules in Chinese Children with Attention-Deficit/Hyperactivity Disorder.

CNS drugs·2026

Assessment of Excised and Reconstructed Human Pigmented Skin Models for In Vitro Permeation Testing.

European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences·2026

Development of orodispersible wafer-based delayed-release omeprazole systems for pediatric compounding.

International journal of pharmaceutics·2026

Common Deficiencies in Dossiers of Finished Pharmaceutical Products Submitted for Registration and Related Factors: A Mixed-Method Study in Tanzania.

Therapeutic innovation & regulatory science·2026

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Lead development: validation and application of high throughput screening for determination of pharmacokinetic

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Induction of spermatogenesis by androgens in gonadotropin-deficient (hpg) mice.

Dysfibrinogenemia: a case with thrombosis (fibrinogen Richfield) and an overview of the clinical and laboratory spectrum.

Purification and properties of four monocot lectins from the family Araceae.

Concurrent evaluation of immunization programme by Lot Quality Assurance Sampling.

Characterization of a low-temperature-induced cDNA from winter Brassica napus encoding the 70 kDa subunit of tonoplast ATPase.

Structural studies on the PH domains of Db1, Sos1, IRS-1, and beta ARK1 and their differential binding to G beta gamma subunits.

Synthesis of axially chiral benzochalcogenophene derivatives and their anti-proliferative activities in cancer cells.

Hypoxia-activated 2-nitroimidazole-brusatol carbonate prodrugs for enhanced gastric cancer therapy with reduced systemic toxicity.

Rivastigmine-centered molecular hybridization strategies for multi-targeted intervention in Alzheimer's disease: Advances (2020-2026).

Criteria-guided selection of alternative zinc-binding groups of HDAC3 inhibitors using in silico and in vitro approaches.

Design, synthesis, and biological evaluation of novel dihydropyrimidinone imines as potent anticancer agents targeting AKT to induce cell cycle arrest and apoptosis in breast Cancer cells.

Design, synthesis, biological and computational evaluation of Thieno[3,2-d]pyrimidine-based inhibitors of JAK3 kinase.

Quantification of PDGF-AB and TGF-β1 Proteins in Platelet-rich Plasma Obtained under Different Conditions.

A Multiparametric in vitro Strategy for Small Molecule Drug-Induced Liver Injury Risk Mitigation in Early Drug Development.

A Phase 3, Multicenter, Randomized, Placebo-Controlled Trial Evaluating the Efficacy, Safety, and Tolerability of Serdexmethylphenidate/d-Methylphenidate Capsules in Chinese Children with Attention-Deficit/Hyperactivity Disorder.

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Development of orodispersible wafer-based delayed-release omeprazole systems for pediatric compounding.

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Lead development: validation and application of high throughput screening for determination of pharmacokinetic...

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Lead development: validation and application of high throughput screening for determination of pharmacokinetic