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Preparation of Stable Bicyclic Aziridinium Ions and Their Ring-Opening for the Synthesis of Azaheterocycles
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5-(Piperidin-2-yl)- and 5-(homopiperidin-2-yl)-1,4-benzodiazepines: high-affinity, basic ligands for the

J L Castro1, H B Broughton, M G Russell

  • 1Chemistry Department, Merck Sharp & Dohme Research Laboratories, Harlow, Essex, U.K.

Journal of Medicinal Chemistry
|August 1, 1997
PubMed

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