SR141716A is an inverse agonist at the human cannabinoid CB1 receptor

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Updated: Oct 31, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
07:41

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

Published on: February 20, 2018

R S Landsman1, T H Burkey, P Consroe

  • 1Department of Pharmacology, University of Arizona Health Sciences Center, Tucson 85724, USA.

European Journal of Pharmacology
|November 5, 1997
PubMed

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