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[Antimicrobial activities of clindamycin against clinical isolated Streptococcus pneumoniae]

Y Suzuki1, R Ishihara, Y Ishii

  • 1Section of Studies, Tokyo Clinical Research Center.

Insights

Clindamycin (CLDM) demonstrates potent activity against macrolide (MLs)-inducible resistant Streptococcus pneumoniae strains, particularly those resistant to penicillin. Susceptibility testing for CLDM is recommended when S. pneumoniae is detected.

Area of Science:

  • Microbiology
  • Infectious Diseases
  • Pharmacology

Background:

  • Macrolide resistance in Streptococcus pneumoniae is a growing clinical concern.
  • Penicillin-intermediate and resistant strains exhibit high rates of macrolide resistance.
  • Understanding resistance mechanisms is crucial for effective antibiotic therapy.

Purpose of the Study:

  • To evaluate the in vitro antimicrobial activity of clindamycin (CLDM) against clinical isolates of Streptococcus pneumoniae.
  • To assess CLDM's efficacy against macrolide-resistant S. pneumoniae strains, considering different penicillin susceptibility profiles.
  • To determine the prevalence of inducible and constitutive macrolide resistance mechanisms.

Main Methods:

  • Antimicrobial susceptibility testing of S. pneumoniae isolates using clindamycin.
  • Determination of minimum inhibitory concentration (MIC70) values for CLDM.
  • Classification of isolates based on penicillin susceptibility (PSSP, PISP, PRSP) and macrolide resistance phenotype (inducible vs. constitutive).

Main Results:

  • High frequencies of macrolide resistance were observed in penicillin-intermediate/resistant S. pneumoniae (92.0%) compared to susceptible strains (48.0%).
  • MLs-inducible resistance was more prevalent in PISP/PRSP (66.0%) than PSSP (24.6%), while MLs-constitutive resistance was more frequent in PSSP (24.0%).
  • Clindamycin exhibited strong activity against MLs-inducible resistant strains (MIC70 ≤ 0.025 µg/ml for PSSP, 0.1 µg/ml for PISP/PRSP), but weak activity against MLs-constitutive resistant strains.

Conclusions:

  • Clindamycin is effective against macrolide-inducible resistant Streptococcus pneumoniae, especially penicillin-intermediate/resistant strains.
  • The high prevalence of inducible resistance in PISP/PRSP suggests clindamycin as a potential therapeutic option.
  • Antimicrobial susceptibility testing for clindamycin is recommended for all S. pneumoniae infections to guide treatment decisions.

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