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Inhibition of inducible nitric oxide synthase after myocardial ischemia increases coronary flow

P E Parrino1, V E Laubach, J R Gaughen

  • 1Department of Surgery, University of Virginia Health Sciences Center, Charlottesville 22908, USA.

Abstract

Insights

Selective inhibition of inducible nitric oxide synthase significantly increased coronary flow after ischemia. This effect was observed with reduced neutrophil accumulation and improved contractility, highlighting its role in myocardial ischemia-reperfusion injury.

Area of Science:

  • Cardiovascular Physiology
  • Biomedical Research
  • Pharmacology

Background:

  • Nitric oxide synthase (NOS) plays a complex role in myocardial ischemia-reperfusion (I/R) injury.
  • Inducible nitric oxide synthase (iNOS) is hypothesized to regulate coronary blood flow post-ischemia.

Purpose of the Study:

  • To investigate the role of iNOS in regulating coronary blood flow following myocardial ischemia.
  • To assess the impact of iNOS inhibition on cardiac function and inflammatory markers during I/R.

Main Methods:

  • Isolated blood-perfused rabbit hearts subjected to ischemia-reperfusion protocols.
  • Treatment with N omega-nitro-L-arginine methyl ester (L-NAME) or the selective iNOS inhibitor 1400W during reperfusion.
  • Measurement of left ventricular developed pressure, coronary flow, myeloperoxidase, and cyclic guanosine monophosphate.

Main Results:

  • Selective iNOS inhibition with 1400W significantly increased coronary flow post-ischemia compared to L-NAME and control.
  • No significant differences in left ventricular developed pressure or cyclic guanosine monophosphate levels were observed among ischemic groups.
  • Myeloperoxidase levels were elevated in L-NAME treated hearts, indicating reduced neutrophil accumulation with 1400W.

Conclusions:

  • Highly selective iNOS inhibition enhances coronary flow post-ischemia, independent of cyclic guanosine monophosphate levels.
  • This inhibition is associated with decreased neutrophil infiltration and a trend toward improved contractility.
  • iNOS plays a critical role in modulating coronary blood flow dynamics during myocardial I/R injury.

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