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Efficacious, orally bioavailable thrombin inhibitors based on 3-aminopyridinone or 3-aminopyrazinone acetamide

P E Sanderson1, T A Lyle, K J Cutrona

  • 1Departments of Antiviral Research, Biological Chemistry, Drug Metabolism, Medicinal Chemistry, Molecular Design and Diversity, Pharmacology, Merck Research Laboratories, West Point, Pennsylvania 19486, USA.

Journal of Medicinal Chemistry
|November 7, 1998
PubMed

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