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Chemical Biology & Drug Design|March 13, 2012
A combined study using ligand-based design, synthesis, and pharmacological evaluation of analogues of the acetaminophen ortho-regioisomer with potent analgesic activityLuana M D Queiroz, Josmar R Rocha, Andrei Leitão, et al.Medicinal Chemistry (Shariqah (United Arab Emirates))|May 14, 2015
Molecular design, synthesis and evaluation of 2,3-diarylquinoxalines as estrogen receptor ligandsDiego P Sangi, Márcia R Cominetti, Amanda B Becceneri, et al.Anti-Cancer Agents in Medicinal Chemistry|October 30, 2018
Biological Activity and Physicochemical Properties of Dipeptidyl Nitrile Derivatives Against Pancreatic Ductal Adenocarcinoma CellsJosé C Quilles, Murillo D L Bernardi, Pedro H J Batista, et al.RSC Advances|May 11, 2022
Apoferritin encapsulation of cysteine protease inhibitors for cathepsin L inhibition in cancer cellsJosé C Quilles Junior, Fernanda Dos Reis Rocho Carlos, A Montanari, et al.Journal of Computer-Aided Molecular Design|November 26, 2003
3D QSAR studies on binding affinities of coumarin natural products for glycosomal GAPDH of Trypanosoma cruziIrwin R A Menezes, Julio C D Lopes, Carlos A Montanari, et al.ACS Medicinal Chemistry Letters|July 26, 2017
New Class of Antitrypanosomal Agents Based on ImidazopyridinesDaniel G Silva, J Robert Gillespie, Ranae M Ranade, et al.Journal of Chemical Information and Modeling|August 31, 2022
Assessment of Reversibility for Covalent Cysteine Protease Inhibitors Using Quantum Mechanics/Molecular Mechanics Free Energy SurfacesAlberto M Dos Santos, Amanda Ruslana Santana Oliveira, Clauber H S da Costa, et al.Bioorganic & Medicinal Chemistry Letters|August 9, 2020
N-Sulfonyl dipeptide nitriles as inhibitors of human cathepsin S: In silico design, synthesis and biochemical characterizationCarina Lemke, Lorenzo Cianni, Christian Feldmann, et al.Bioorganic & Medicinal Chemistry|March 4, 2009
Discovery of novel Trypanosoma cruzi glyceraldehyde-3-phosphate dehydrogenase inhibitorsRenato F Freitas, Igor M Prokopczyk, Aderson Zottis, et al.Current Topics in Medicinal Chemistry|March 26, 2014
Structure based design, synthesis, and evaluation of potential inhibitors of steroid sulfataseE V Costa, E Sousa, K Choosang, et al.Pageof 36