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Journal of Medicinal Chemistry|January 28, 2017
Accepting the Invitation to Open Innovation in Malaria Drug Discovery: Synthesis, Biological Evaluation, and Investigation on the Structure-Activity Relationships of Benzo[b]thiophene-2-carboxamides as Antimalarial AgentsMarco Pieroni, Elisa Azzali, Nicoletta Basilico, et al.Biotechnology and Applied Biochemistry|September 7, 2017
Membrane cholesterol effect on the 5-HT<sub>2A</sub> receptor: Insights into the lipid-induced modulation of an antipsychotic drug targetJuan Manuel Ramírez-Anguita, Ismael Rodríguez-Espigares, Ramon Guixà-González, et al.Proteins|September 8, 2021
Crystal structure of Aspergillus fumigatus AroH, an aromatic amino acid aminotransferaseSharon Spizzichino, Gioena Pampalone, Mirco Dindo, et al.Journal of Molecular Graphics & Modelling|March 15, 2019
Pharmacophore modeling and virtual screening studies to identify novel selective SIRT2 inhibitorsGokcen Eren, Agostino Bruno, Sezen Guntekin-Ergun, et al.Frontiers in Molecular Biosciences|December 15, 2018
Biochemical Characterization of <i>Aspergillus fumigatus</i> AroH, a Putative Aromatic Amino Acid AminotransferaseMirco Dindo, Egidia Costanzi, Marco Pieroni, et al.Chemmedchem|June 16, 2016
Discovery of New Potential Anti-Infective Compounds Based on Carbonic Anhydrase Inhibitors by Rational Target-Focused Repurposing ApproachesGiannamaria Annunziato, Andrea Angeli, Francesca D'Alba, et al.ACS Chemical Neuroscience|July 4, 2019
Unbinding of Translocator Protein 18 kDa (TSPO) Ligands: From in Vitro Residence Time to in Vivo Efficacy via in Silico SimulationsAgostino Bruno, Elisabetta Barresi, Nicola Simola, et al.Chemmedchem|May 19, 2017
Identification of Breast Cancer Inhibitors Specific for G Protein-Coupled Estrogen Receptor (GPER)-Expressing CellsFrancesca Aiello, Gabriele Carullo, Francesca Giordano, et al.ACS Medicinal Chemistry Letters|May 22, 2020
Inhibition of Nonessential Bacterial Targets: Discovery of a Novel Serine <i>O</i>-Acetyltransferase InhibitorJoana Magalhães, Nina Franko, Samanta Raboni, et al.Journal of Enzyme Inhibition and Medicinal Chemistry|September 1, 2016
Cyclopropane-1,2-dicarboxylic acids as new tools for the biophysical investigation of O-acetylserine sulfhydrylases by fluorimetric methods and saturation transfer difference (STD) NMRGiannamaria Annunziato, Marco Pieroni, Roberto Benoni, et al.Pageof 8