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Analytical Biochemistry|December 29, 2023
Proficiently partitioning of bioactive peptide-ssDNA conjugates by microbead-assisted capillary electrophoresis (MACE)Muneyuki Matsuo, Koji Wakui, Yuuki Inami, et al.Bioorganic & Medicinal Chemistry Letters|December 26, 2008
(-)-Cercosporamide derivatives as novel antihyperglycemic agentsAkihiro Furukawa, Tsuyoshi Arita, Susumu Satoh, et al.Bioorganic & Medicinal Chemistry|February 21, 2018
CycLS: Accurate, whole-library sequencing of cyclic peptides using tandem mass spectrometryChad Townsend, Akihiro Furukawa, Joshua Schwochert, et al.Journal of Medicinal Chemistry|October 4, 2016
Passive Membrane Permeability in Cyclic Peptomer Scaffolds Is Robust to Extensive Variation in Side Chain Functionality and Backbone GeometryAkihiro Furukawa, Chad E Townsend, Joshua Schwochert, et al.Bioorganic & Medicinal Chemistry Letters|March 12, 2010
Discovery of a novel selective PPARgamma modulator from (-)-Cercosporamide derivativesAkihiro Furukawa, Tsuyoshi Arita, Susumu Satoh, et al.Bioorganic & Medicinal Chemistry Letters|January 10, 2012
Substituents at the naphthalene C3 position of (-)-Cercosporamide derivatives significantly affect the maximal efficacy as PPARγ partial agonistsAkihiro Furukawa, Tsuyoshi Arita, Takehiro Fukuzaki, et al.Angewandte Chemie (International Ed. in English)|August 14, 2020
Drug-Like Properties in Macrocycles above MW 1000: Backbone Rigidity versus Side-Chain LipophilicityAkihiro Furukawa, Joshua Schwochert, Cameron R Pye, et al.Biological & Pharmaceutical Bulletin|July 2, 2011
Pharmacology and in vitro profiling of a novel peroxisome proliferator-activated receptor γ ligand, Cerco-AKenji Wakabayashi, Shinko Hayashi, Yumi Matsui, et al.European Journal of Medicinal Chemistry|June 26, 2012
Synthesis and biological evaluation of novel (-)-Cercosporamide derivatives as potent selective PPARγ modulatorsAkihiro Furukawa, Tsuyoshi Arita, Takehiro Fukuzaki, et al.Journal of Medicinal Chemistry|January 7, 2017
Nonclassical Size Dependence of Permeation Defines Bounds for Passive Adsorption of Large Drug MoleculesCameron R Pye, William M Hewitt, Joshua Schwochert, et al.Pageof 2