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Current Medicinal Chemistry|June 2, 2026
Design, Synthesis, and Pharmacological Characterization of Substituted Quinoxalines as NOP Receptor LigandsDonald J Kyle, Naoki Tsuno, Laykea Tafesse, et al.Journal of Medicinal Chemistry|July 25, 2014
Structure-activity relationship studies and discovery of a potent transient receptor potential vanilloid (TRPV1) antagonist 4-[3-chloro-5-[(1S)-1,2-dihydroxyethyl]-2-pyridyl]-N-[5-(trifluoromethyl)-2-pyridyl]-3,6-dihydro-2H-pyridine-1-carboxamide (V116517) as a clinical candidate for pain managementLaykea Tafesse, Toshiyuki Kanemasa, Noriyuki Kurose, et al.Cancer Immunology Research|January 30, 2016
CAR T Cells Targeting Podoplanin Reduce Orthotopic Glioblastomas in Mouse BrainsSatoshi Shiina, Masasuke Ohno, Fumiharu Ohka, et al.Science Advances|February 20, 2026
Glomerular routing of tumor-derived extracellular vesicles substantiates urinary biopsyShota Kawaguchi, Taiga Ajiri, Rina Mitsuya, et al.Nature Communications|December 5, 2022
Pexophagy suppresses ROS-induced damage in leaf cells under high-intensity lightKazusato Oikawa, Shino Goto-Yamada, Yasuko Hayashi, et al.Human Molecular Genetics|December 1, 2006
The DYRK1A gene, encoded in chromosome 21 Down syndrome critical region, bridges between beta-amyloid production and tau phosphorylation in Alzheimer diseaseRyo Kimura, Kouzin Kamino, Mitsuko Yamamoto, et al.Neuro-Oncology|July 2, 2021
Newly established patient-derived organoid model of intracranial meningiomaShintaro Yamazaki, Fumiharu Ohka, Masaki Hirano, et al.Acta Neuropathologica Communications|February 6, 2020
H3F3A mutant allele specific imbalance in an aggressive subtype of diffuse midline glioma, H3 K27M-mutantSachi Maeda, Fumiharu Ohka, Yusuke Okuno, et al.Journal of Medicinal Chemistry|February 16, 2021
Discovery of Atabecestat (JNJ-54861911): A Thiazine-Based β-Amyloid Precursor Protein Cleaving Enzyme 1 Inhibitor Advanced to the Phase 2b/3 EARLY Clinical TrialYuji Koriyama, Akihiro Hori, Hisanori Ito, et al.Journal of Neurochemistry|November 7, 2006
BACE1 inhibition reduces endogenous Abeta and alters APP processing in wild-type miceKouhei Nishitomi, Gaku Sakaguchi, Yuko Horikoshi, et al.Pageof 19