Jove
Visualize
Contact Us
JoVE
x logofacebook logolinkedin logoyoutube logo
ABOUT JoVE
OverviewLeadershipBlogJoVE Help Center
AUTHORS
Publishing ProcessEditorial BoardScope & PoliciesPeer ReviewFAQSubmit
LIBRARIANS
TestimonialsSubscriptionsAccessResourcesLibrary Advisory BoardFAQ
RESEARCH
JoVE JournalMethods CollectionsJoVE Encyclopedia of ExperimentsArchive
EDUCATION
JoVE CoreJoVE BusinessJoVE Science EducationJoVE Lab ManualFaculty Resource CenterFaculty Site
Terms & Conditions of Use
Privacy Policy
Policies

Filters

Aleem Gangjee

Showing results (61-70 of 132) with videos related to

Pageof 14
Sort By:
Biochemical Pharmacology|June 9, 2004
Inhibition of insulin-like growth factor I receptor autophosphorylation by novel 6-5 ring-fused compoundsWanqing Li, Svetlana Favelyukis, Jie Yang, et al.
Journal of Medicinal Chemistry|May 1, 2013
Design, synthesis, and molecular modeling of novel pyrido[2,3-d]pyrimidine analogues as antifolates; application of Buchwald-Hartwig aminations of heterocyclesAleem Gangjee, Ojas A Namjoshi, Sudhir Raghavan, et al.
Biochemistry|February 11, 2017
Correction to Structural and Enzymatic Analysis of Tumor-Targeted Antifolates That Inhibit Glycinamide Ribonucleotide FormyltransferaseSiobhan M Deis, Arpit Doshi, Zhanjun Hou, et al.
The Biochemical Journal|March 28, 2019
Regulation of differential proton-coupled folate transporter gene expression in human tumors: transactivation by KLF15 with NRF-1 and the role of Sp1Zhanjun Hou, Carrie O'Connor, Josephine Frühauf, et al.
Journal of Medicinal Chemistry|February 7, 2003
Design, synthesis, and biological activities of classical N-[4-[2-(2-amino-4-ethylpyrrolo[2,3-d]pyrimidin-5-yl)ethyl]benzoyl]-l-glutamic acid and its 6-methyl derivative as potential dual inhibitors of thymidylate synthase and dihydrofolate reductase and as potential antitumor agentsAleem Gangjee, Jianming Yu, Roy L Kisliuk, et al.
Bioorganic & Medicinal Chemistry|November 5, 2019
Discovery of amide-bridged pyrrolo[2,3-d]pyrimidines as tumor targeted classical antifolates with selective uptake by folate receptor α and inhibition of de novo purine nucleotide biosynthesisWeiguo Xiang, Aamod Dekhne, Arpit Doshi, et al.
Molecular Pharmacology|January 10, 2008
Role of lysine 411 in substrate carboxyl group binding to the human reduced folate carrier, as determined by site-directed mutagenesis and affinity inhibitionYijun Deng, Zhanjun Hou, Lei Wang, et al.
Journal of Medicinal Chemistry|January 17, 2012
Synthesis and biological activity of 6-substituted pyrrolo[2,3-d]pyrimidine thienoyl regioisomers as inhibitors of de novo purine biosynthesis with selectivity for cellular uptake by high affinity folate receptors and the proton-coupled folate transporter over the reduced folate carrierLei Wang, Christina Cherian, Sita Kugel Desmoulin, et al.
BMC Cancer|July 17, 2015
A new anti-glioma therapy, AG119: pre-clinical assessment in a mouse GL261 glioma modelRheal A Towner, Michael Ihnat, Debra Saunders, et al.
Bioorganic & Medicinal Chemistry|November 30, 2016
Discovery and preclinical evaluation of 7-benzyl-N-(substituted)-pyrrolo[3,2-d]pyrimidin-4-amines as single agents with microtubule targeting effects along with triple-acting angiokinase inhibition as antitumor agentsRoheeth Kumar Pavana, Shruti Choudhary, Anja Bastian, et al.
Pageof 14

Showing results (61-70 of 132) with videos related to

Sort By:
Pageof 14
Biochemical Pharmacology|June 9, 2004
Inhibition of insulin-like growth factor I receptor autophosphorylation by novel 6-5 ring-fused compoundsWanqing Li, Svetlana Favelyukis, Jie Yang, et al.
Journal of Medicinal Chemistry|May 1, 2013
Design, synthesis, and molecular modeling of novel pyrido[2,3-d]pyrimidine analogues as antifolates; application of Buchwald-Hartwig aminations of heterocyclesAleem Gangjee, Ojas A Namjoshi, Sudhir Raghavan, et al.
Biochemistry|February 11, 2017
Correction to Structural and Enzymatic Analysis of Tumor-Targeted Antifolates That Inhibit Glycinamide Ribonucleotide FormyltransferaseSiobhan M Deis, Arpit Doshi, Zhanjun Hou, et al.
The Biochemical Journal|March 28, 2019
Regulation of differential proton-coupled folate transporter gene expression in human tumors: transactivation by KLF15 with NRF-1 and the role of Sp1Zhanjun Hou, Carrie O'Connor, Josephine Frühauf, et al.
Journal of Medicinal Chemistry|February 7, 2003
Design, synthesis, and biological activities of classical N-[4-[2-(2-amino-4-ethylpyrrolo[2,3-d]pyrimidin-5-yl)ethyl]benzoyl]-l-glutamic acid and its 6-methyl derivative as potential dual inhibitors of thymidylate synthase and dihydrofolate reductase and as potential antitumor agentsAleem Gangjee, Jianming Yu, Roy L Kisliuk, et al.
Bioorganic & Medicinal Chemistry|November 5, 2019
Discovery of amide-bridged pyrrolo[2,3-d]pyrimidines as tumor targeted classical antifolates with selective uptake by folate receptor α and inhibition of de novo purine nucleotide biosynthesisWeiguo Xiang, Aamod Dekhne, Arpit Doshi, et al.
Molecular Pharmacology|January 10, 2008
Role of lysine 411 in substrate carboxyl group binding to the human reduced folate carrier, as determined by site-directed mutagenesis and affinity inhibitionYijun Deng, Zhanjun Hou, Lei Wang, et al.
Journal of Medicinal Chemistry|January 17, 2012
Synthesis and biological activity of 6-substituted pyrrolo[2,3-d]pyrimidine thienoyl regioisomers as inhibitors of de novo purine biosynthesis with selectivity for cellular uptake by high affinity folate receptors and the proton-coupled folate transporter over the reduced folate carrierLei Wang, Christina Cherian, Sita Kugel Desmoulin, et al.
BMC Cancer|July 17, 2015
A new anti-glioma therapy, AG119: pre-clinical assessment in a mouse GL261 glioma modelRheal A Towner, Michael Ihnat, Debra Saunders, et al.
Bioorganic & Medicinal Chemistry|November 30, 2016
Discovery and preclinical evaluation of 7-benzyl-N-(substituted)-pyrrolo[3,2-d]pyrimidin-4-amines as single agents with microtubule targeting effects along with triple-acting angiokinase inhibition as antitumor agentsRoheeth Kumar Pavana, Shruti Choudhary, Anja Bastian, et al.
Pageof 14