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Alessandro Bonardi

Showing results (61-70 of 109) with videos related to

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Journal of Medicinal Chemistry|June 11, 2020
Sulfonamide Inhibitors of Human Carbonic Anhydrases Designed through a Three-Tails Approach: Improving Ligand/Isoform Matching and Selectivity of ActionAlessandro Bonardi, Alessio Nocentini, Silvia Bua, et al.
European Journal of Medicinal Chemistry|April 24, 2018
Dual-tail arylsulfone-based benzenesulfonamides differently match the hydrophobic and hydrophilic halves of human carbonic anhydrases active sites: Selective inhibitors for the tumor-associated hCA IX isoformHany S Ibrahim, Heba Abdelrasheed Allam, Walaa R Mahmoud, et al.
European Journal of Medicinal Chemistry|April 5, 2025
Repurposing the amino-3,5-dicyanopyridine scaffold from adenosine receptor ligands to carbonic anhydrase activatorsErica Vigiani, Alessandro Bonardi, Daniela Catarzi, et al.
Journal of Enzyme Inhibition and Medicinal Chemistry|March 23, 2023
Synthesis, biological evaluation and theoretical studies of (<i>E</i>)-1-(4-sulfamoyl-phenylethyl)-3-arylidene-5-aryl-1H-pyrrol-2(3H)-ones as human carbonic anhydrase inhibitorsFarhat Ramzan, Syed Ayaz Nabi, Mehak Saba Lone, et al.
Bioorganic Chemistry|March 31, 2023
Arylidine extensions of 3-methyl-5-oxo-4,5-dihydro-1H-pyrazol-benzenesulfonamide derivatives: Synthesis, computational simulations and biological evaluation as tumor-associated carbonic anhydrase inhibitorsHeba M Metwally, Heba Abdelrasheed Allam, Fady Baselious, et al.
European Journal of Medicinal Chemistry|February 12, 2020
Inclusion of a 5-fluorouracil moiety in nitrogenous bases derivatives as human carbonic anhydrase IX and XII inhibitors produced a targeted action against MDA-MB-231 and T47D breast cancer cellsAndrea Petreni, Alessandro Bonardi, Carrie Lomelino, et al.
European Journal of Medicinal Chemistry|October 10, 2020
Novel 3-substituted coumarins as selective human carbonic anhydrase IX and XII inhibitors: Synthesis, biological and molecular dynamics analysisMohamed A Abdelrahman, Hany S Ibrahim, Alessio Nocentini, et al.
Journal of Enzyme Inhibition and Medicinal Chemistry|May 31, 2022
Cloning, purification, kinetic and anion inhibition studies of a recombinant β-carbonic anhydrase from the Atlantic salmon parasite platyhelminth <i>Gyrodactylus salaris</i>Ashok Aspatwar, Harlan Barker, Heidi Aisala, et al.
Journal of Enzyme Inhibition and Medicinal Chemistry|April 20, 2023
Effect of hydrophobic extension of aryl enaminones and pyrazole-linked compounds combined with sulphonamide, sulfaguanidine, or carboxylic acid functionalities on carbonic anhydrase inhibitory potency and selectivityHeba Abdelrasheed Allam, Mohamed E Albakry, Walaa R Mahmoud, et al.
Journal of Medicinal Chemistry|June 7, 2023
6-Substituted Triazolyl Benzoxaboroles as Selective Carbonic Anhydrase Inhibitors: Alessio Nocentini, Alessandro Bonardi, Carla Bazzicalupi, et al.
Pageof 11

Showing results (61-70 of 109) with videos related to

Sort By:
Pageof 11
Journal of Medicinal Chemistry|June 11, 2020
Sulfonamide Inhibitors of Human Carbonic Anhydrases Designed through a Three-Tails Approach: Improving Ligand/Isoform Matching and Selectivity of ActionAlessandro Bonardi, Alessio Nocentini, Silvia Bua, et al.
European Journal of Medicinal Chemistry|April 24, 2018
Dual-tail arylsulfone-based benzenesulfonamides differently match the hydrophobic and hydrophilic halves of human carbonic anhydrases active sites: Selective inhibitors for the tumor-associated hCA IX isoformHany S Ibrahim, Heba Abdelrasheed Allam, Walaa R Mahmoud, et al.
European Journal of Medicinal Chemistry|April 5, 2025
Repurposing the amino-3,5-dicyanopyridine scaffold from adenosine receptor ligands to carbonic anhydrase activatorsErica Vigiani, Alessandro Bonardi, Daniela Catarzi, et al.
Journal of Enzyme Inhibition and Medicinal Chemistry|March 23, 2023
Synthesis, biological evaluation and theoretical studies of (<i>E</i>)-1-(4-sulfamoyl-phenylethyl)-3-arylidene-5-aryl-1H-pyrrol-2(3H)-ones as human carbonic anhydrase inhibitorsFarhat Ramzan, Syed Ayaz Nabi, Mehak Saba Lone, et al.
Bioorganic Chemistry|March 31, 2023
Arylidine extensions of 3-methyl-5-oxo-4,5-dihydro-1H-pyrazol-benzenesulfonamide derivatives: Synthesis, computational simulations and biological evaluation as tumor-associated carbonic anhydrase inhibitorsHeba M Metwally, Heba Abdelrasheed Allam, Fady Baselious, et al.
European Journal of Medicinal Chemistry|February 12, 2020
Inclusion of a 5-fluorouracil moiety in nitrogenous bases derivatives as human carbonic anhydrase IX and XII inhibitors produced a targeted action against MDA-MB-231 and T47D breast cancer cellsAndrea Petreni, Alessandro Bonardi, Carrie Lomelino, et al.
European Journal of Medicinal Chemistry|October 10, 2020
Novel 3-substituted coumarins as selective human carbonic anhydrase IX and XII inhibitors: Synthesis, biological and molecular dynamics analysisMohamed A Abdelrahman, Hany S Ibrahim, Alessio Nocentini, et al.
Journal of Enzyme Inhibition and Medicinal Chemistry|May 31, 2022
Cloning, purification, kinetic and anion inhibition studies of a recombinant β-carbonic anhydrase from the Atlantic salmon parasite platyhelminth <i>Gyrodactylus salaris</i>Ashok Aspatwar, Harlan Barker, Heidi Aisala, et al.
Journal of Enzyme Inhibition and Medicinal Chemistry|April 20, 2023
Effect of hydrophobic extension of aryl enaminones and pyrazole-linked compounds combined with sulphonamide, sulfaguanidine, or carboxylic acid functionalities on carbonic anhydrase inhibitory potency and selectivityHeba Abdelrasheed Allam, Mohamed E Albakry, Walaa R Mahmoud, et al.
Journal of Medicinal Chemistry|June 7, 2023
6-Substituted Triazolyl Benzoxaboroles as Selective Carbonic Anhydrase Inhibitors: Alessio Nocentini, Alessandro Bonardi, Carla Bazzicalupi, et al.
Pageof 11