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Archiv Der Pharmazie
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December 17, 2024
New 7-hydroxycoumarin acetamide derivatives as human carbonic anhydrase IX and XII inhibitors: Design, synthesis, biological evaluation and molecular docking studies
Sarvan Maddipatla, Bulti Bakchi, Mayura Anil Shinde, et al.
European Journal of Medicinal Chemistry
|
December 17, 2021
2-(2-Hydroxyethyl)piperazine derivatives as potent human carbonic anhydrase inhibitors: Synthesis, enzyme inhibition, computational studies and antiglaucoma activity
Niccolò Chiaramonte, Andrea Angeli, Silvia Sgambellone, et al.
Journal of Enzyme Inhibition and Medicinal Chemistry
|
March 21, 2022
The three-tails approach as a new strategy to improve selectivity of action of sulphonamide inhibitors against tumour-associated carbonic anhydrase IX and XII
Alessandro Bonardi, Silvia Bua, Jacob Combs, et al.
International Journal of Molecular Sciences
|
November 13, 2021
Selective Inhibition of <i>Helicobacter pylori</i> Carbonic Anhydrases by Carvacrol and Thymol Could Impair Biofilm Production and the Release of Outer Membrane Vesicles
Rossella Grande, Simone Carradori, Valentina Puca, et al.
European Journal of Medicinal Chemistry
|
November 14, 2019
Synthesis, biological and molecular dynamics investigations with a series of triazolopyrimidine/triazole-based benzenesulfonamides as novel carbonic anhydrase inhibitors
Mohamed A Said, Wagdy M Eldehna, Alessio Nocentini, et al.
Journal of Medicinal Chemistry
|
February 1, 2024
Synthetic Approaches to Novel Human Carbonic Anhydrase Isoform Inhibitors Based on Pyrrol-2-one Moiety
Cristina M Al-Matarneh, Mariana Pinteala, Alina Nicolescu, et al.
Bioorganic Chemistry
|
December 13, 2024
Damsin and neoambrosin: Two sesquiterpene lactones with affinity and different activity for PPAR and TRPA1 receptors
Shymaa I A Abdel-Dayem, Asmaa M Otify, Fabio Arturo Iannotti, et al.
Journal of Medicinal Chemistry
|
May 22, 2024
Development of Penicillin-Based Carbonic Anhydrase Inhibitors Targeting Multidrug-Resistant <i>Neisseria gonorrhoeae</i>
Alessandro Bonardi, Alessio Nocentini, Simone Giovannuzzi, et al.
International Journal of Molecular Sciences
|
May 30, 2019
Novel Diamide-Based Benzenesulfonamides as Selective Carbonic Anhydrase IX Inhibitors Endowed with Antitumor Activity: Synthesis, Biological Evaluation and In Silico Insights
Mohamed A Abdelrahman, Wagdy M Eldehna, Alessio Nocentini, et al.
Archiv Der Pharmazie
|
February 23, 2026
Sideroxylonal B: A Dimeric Phloroglucinol From Eucalyptus cinerea With In Vitro Carbonic Anhydrase Inhibition and Evaluation of Cytotoxicity and Antiviral Potential
Fatema R Saber, Alessandro Bonardi, Rasha A Hassan, et al.
Page
of 11
Search research articles
Search
Showing results (81-90 of 109) with videos related to
Sort By:
Page
of 11
Archiv Der Pharmazie
|
December 17, 2024
New 7-hydroxycoumarin acetamide derivatives as human carbonic anhydrase IX and XII inhibitors: Design, synthesis, biological evaluation and molecular docking studies
Sarvan Maddipatla, Bulti Bakchi, Mayura Anil Shinde, et al.
European Journal of Medicinal Chemistry
|
December 17, 2021
2-(2-Hydroxyethyl)piperazine derivatives as potent human carbonic anhydrase inhibitors: Synthesis, enzyme inhibition, computational studies and antiglaucoma activity
Niccolò Chiaramonte, Andrea Angeli, Silvia Sgambellone, et al.
Journal of Enzyme Inhibition and Medicinal Chemistry
|
March 21, 2022
The three-tails approach as a new strategy to improve selectivity of action of sulphonamide inhibitors against tumour-associated carbonic anhydrase IX and XII
Alessandro Bonardi, Silvia Bua, Jacob Combs, et al.
International Journal of Molecular Sciences
|
November 13, 2021
Selective Inhibition of <i>Helicobacter pylori</i> Carbonic Anhydrases by Carvacrol and Thymol Could Impair Biofilm Production and the Release of Outer Membrane Vesicles
Rossella Grande, Simone Carradori, Valentina Puca, et al.
European Journal of Medicinal Chemistry
|
November 14, 2019
Synthesis, biological and molecular dynamics investigations with a series of triazolopyrimidine/triazole-based benzenesulfonamides as novel carbonic anhydrase inhibitors
Mohamed A Said, Wagdy M Eldehna, Alessio Nocentini, et al.
Journal of Medicinal Chemistry
|
February 1, 2024
Synthetic Approaches to Novel Human Carbonic Anhydrase Isoform Inhibitors Based on Pyrrol-2-one Moiety
Cristina M Al-Matarneh, Mariana Pinteala, Alina Nicolescu, et al.
Bioorganic Chemistry
|
December 13, 2024
Damsin and neoambrosin: Two sesquiterpene lactones with affinity and different activity for PPAR and TRPA1 receptors
Shymaa I A Abdel-Dayem, Asmaa M Otify, Fabio Arturo Iannotti, et al.
Journal of Medicinal Chemistry
|
May 22, 2024
Development of Penicillin-Based Carbonic Anhydrase Inhibitors Targeting Multidrug-Resistant <i>Neisseria gonorrhoeae</i>
Alessandro Bonardi, Alessio Nocentini, Simone Giovannuzzi, et al.
International Journal of Molecular Sciences
|
May 30, 2019
Novel Diamide-Based Benzenesulfonamides as Selective Carbonic Anhydrase IX Inhibitors Endowed with Antitumor Activity: Synthesis, Biological Evaluation and In Silico Insights
Mohamed A Abdelrahman, Wagdy M Eldehna, Alessio Nocentini, et al.
Archiv Der Pharmazie
|
February 23, 2026
Sideroxylonal B: A Dimeric Phloroglucinol From Eucalyptus cinerea With In Vitro Carbonic Anhydrase Inhibition and Evaluation of Cytotoxicity and Antiviral Potential
Fatema R Saber, Alessandro Bonardi, Rasha A Hassan, et al.
Page
of 11