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Bioorganic Chemistry|May 30, 2026
Rationally optimized mucroporin-M1 peptides disrupt viral envelopes and resist degradationClaudia Storti, Annagiulia Favaro, Sara Tuci, et al.European Journal of Medicinal Chemistry|March 4, 2026
Discovery of a tetrahydrobenzothiophen-2-yl-pyrazolo[1,5-a]pyrimidine-3-carboxamide-based PROTAC as degrader of SARS-CoV-2 main proteaseMichela Eleuteri, Alessandro Bazzacco, Beatrice Mercorelli, et al.Chemmedchem|May 23, 2026
Streamlined Synthesis and Structure-Activity Relationship Analysis of 2-Amidothiophene-3-Carboxamides Targeting Influenza Polymerase PA-PB1 HeterodimerizationTommaso Felicetti, Alessia Zago, Andrea Astolfi, et al.Antiviral Research|August 8, 2024
Synergistic activity of an RNA polymerase PA-PB1 interaction inhibitor with oseltamivir against human and avian influenza viruses in cell culture and in ovoAnna Bonomini, Jiwei Zhang, Han Ju, et al.Pageof 1