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Biochemistry|October 1, 2014
Binding hotspots of BAZ2B bromodomain: Histone interaction revealed by solution NMR driven dockingFleur M Ferguson, David M Dias, João P G L M Rodrigues, et al.Cell Chemical Biology|July 16, 2020
Inducible Degradation of Target Proteins through a Tractable Affinity-Directed Protein Missile SystemLuke M Simpson, Thomas J Macartney, Alice Nardin, et al.Molecular Biosystems|August 2, 2011
Bromodomain-peptide displacement assays for interactome mapping and inhibitor discoveryMartin Philpott, Jing Yang, Tony Tumber, et al.European Journal of Pharmacology|May 29, 2018
Identification of compounds acting as negative allosteric modulators of the LPA1 receptorJonathan Ellery, Louise Dickson, Toni Cheung, et al.Journal of Medicinal Chemistry|December 6, 2013
Targeting low-druggability bromodomains: fragment based screening and inhibitor design against the BAZ2B bromodomainFleur M Ferguson, Oleg Fedorov, Apirat Chaikuad, et al.Journal of Medicinal Chemistry|September 14, 2023
Expanding the Structural Diversity at the Phenylene Core of Ligands for the von Hippel-Lindau E3 Ubiquitin Ligase: Development of Highly Potent Hypoxia-Inducible Factor-1α StabilizersLan Phuong Vu, Claudia J Diehl, Ryan Casement, et al.Chemmedchem|June 11, 2021
The 2nd Alpine Winter Conference on Medicinal and Synthetic ChemistryAlessio Ciulli, Lawrence Hamann, Wolfgang Jahnke, et al.Chemmedchem|August 30, 2022
Discovery of Benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First BromodomainAlessandra Cipriano, Ciro Milite, Alessandra Feoli, et al.Journal of the American Chemical Society|November 28, 2024
Leveraging Dual-Ligase Recruitment to Enhance Protein Degradation via a Heterotrivalent Proteolysis Targeting ChimeraAdam G Bond, Miquel Muñoz I Ordoño, Celia M Bisbach, et al.The Biochemical Journal|March 18, 2011
Structural investigation of inhibitor designs targeting 3-dehydroquinate dehydratase from the shikimate pathway of Mycobacterium tuberculosisMarcio V B Dias, William C Snee, Karen M Bromfield, et al.Pageof 16