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European Journal of Medicinal Chemistry|June 20, 2021
Investigation of 3-sulfamoyl coumarins against cancer-related IX and XII isoforms of human carbonic anhydrase as well as cancer cells leads to the discovery of 2-oxo-2H-benzo[h]chromene-3-sulfonamide - A new caspase-activating proapoptotic agentDmitry Dar'in, Grigory Kantin, Stanislav Kalinin, et al.Chemmedchem|August 4, 2020
Synthesis, Computational Studies and Assessment of in Vitro Activity of Squalene Derivatives as Carbonic Anhydrase InhibitorsLilia Clima, Bogdan Florin Craciun, Andrea Angeli, et al.Journal of Enzyme Inhibition and Medicinal Chemistry|October 31, 2019
Phosphonamidates are the first phosphorus-based zinc binding motif to show inhibition of β-class carbonic anhydrases from bacteria, fungi, and protozoaSiham A Alissa, Hanan A Alghulikah, Zeid A Alothman, et al.Chemmedchem|April 21, 2026
A New Series of Amino Alcohol Oxime Ethers as Activators of Human Brain Carbonic Anhydrases: Advances in Selective Activation of Human Carbonic Anhydrase VIICamilla Mangini, Riccardo Di Leo, Jacopo Castagnoli, et al.Journal of Enzyme Inhibition and Medicinal Chemistry|October 18, 2023
Design, synthesis, and biological investigation of selective human carbonic anhydrase II, IX, and XII inhibitors using 7-aryl/heteroaryl triazolopyrimidines bearing a sulfanilamide scaffoldRomeo Romagnoli, Tiziano De Ventura, Stefano Manfredini, et al.Journal of Enzyme Inhibition and Medicinal Chemistry|December 21, 2019
Inhibition survey with phenolic compounds against the δ- and η-class carbonic anhydrases from the marine diatom thalassiosira weissflogii and protozoan Plasmodium falciparumSiham A Alissa, Hanan A Alghulikah, Zeid A ALOthman, et al.Bioorganic & Medicinal Chemistry|March 28, 2017
Inhibition of Malassezia globosa carbonic anhydrase with phenolsYeganeh Entezari Heravi, Silvia Bua, Alessio Nocentini, et al.Journal of Enzyme Inhibition and Medicinal Chemistry|April 19, 2022
Novel 3-(6-methylpyridin-2-yl)coumarin-based chalcones as selective inhibitors of cancer-related carbonic anhydrases IX and XII endowed with anti-proliferative activityHaytham O Tawfik, Moataz A Shaldam, Alessio Nocentini, et al.Journal of Medicinal Chemistry|January 19, 2026
Targeting Metabolic and pH Regulatory Pathways in Cancer via Dual Inhibition of Nicotinamide Phosphoribosyltransferase and Carbonic Anhydrases IX and XIINiccolò Paoletti, Simone Giovannuzzi, Massimiliano Gasparrini, et al.International Journal of Molecular Sciences|January 23, 2024
Leveraging SARS-CoV-2 Main Protease (Mpro) for COVID-19 Mitigation with Selenium-Based InhibitorsViviana De Luca, Andrea Angeli, Alessio Nocentini, et al.Pageof 29