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Bioorganic Chemistry|April 13, 2019
Novel synthesized SLC-0111 thiazole and thiadiazole analogues: Determination of their carbonic anhydrase inhibitory activity and molecular modeling studiesMahmoud F Abo-Ashour, Wagdy M Eldehna, Alessio Nocentini, et al.Journal of Enzyme Inhibition and Medicinal Chemistry|August 3, 2017
Inhibition of the β-carbonic anhydrase from the dandruff-producing fungus Malassezia globosa with monothiocarbamatesAlessio Nocentini, Daniela Vullo, Sonia Del Prete, et al.International Journal of Biological Macromolecules|August 28, 2024
Discovery of new sulfonamide-tethered 2-aryl-4-anilinoquinazolines as the first-in-class dual carbonic anhydrase and EGFR inhibitorsWagdy M Eldehna, Zainab M Elsayed, Andrea Ammara, et al.European Journal of Medicinal Chemistry|February 12, 2020
Inclusion of a 5-fluorouracil moiety in nitrogenous bases derivatives as human carbonic anhydrase IX and XII inhibitors produced a targeted action against MDA-MB-231 and T47D breast cancer cellsAndrea Petreni, Alessandro Bonardi, Carrie Lomelino, et al.Chemmedchem|March 26, 2018
Natural Polyphenols Selectively Inhibit β-Carbonic Anhydrase from the Dandruff-Producing Fungus Malassezia globosa: Activity and Modeling StudiesAlessio Nocentini, Silvia Bua, Sonia Del Prete, et al.Journal of Medicinal Chemistry|June 11, 2020
Sulfonamide Inhibitors of Human Carbonic Anhydrases Designed through a Three-Tails Approach: Improving Ligand/Isoform Matching and Selectivity of ActionAlessandro Bonardi, Alessio Nocentini, Silvia Bua, et al.Molecules (Basel, Switzerland)|May 24, 2020
Hypoxia-Activated Prodrug Derivatives of Carbonic Anhydrase Inhibitors in Benzenesulfonamide Series: Synthesis and Biological EvaluationEmilie Anduran, Ashok Aspatwar, Nanda-Kumar Parvathaneni, et al.European Journal of Medicinal Chemistry|April 24, 2018
Dual-tail arylsulfone-based benzenesulfonamides differently match the hydrophobic and hydrophilic halves of human carbonic anhydrases active sites: Selective inhibitors for the tumor-associated hCA IX isoformHany S Ibrahim, Heba Abdelrasheed Allam, Walaa R Mahmoud, et al.European Journal of Medicinal Chemistry|March 28, 2021
Insertion of metal carbenes into the anilinic N-H bond of unprotected aminobenzenesulfonamides delivers low nanomolar inhibitors of human carbonic anhydrase IX and XII isoformsTatiana Sharonova, Polina Paramonova, Stanislav Kalinin, et al.European Journal of Medicinal Chemistry|April 5, 2025
Repurposing the amino-3,5-dicyanopyridine scaffold from adenosine receptor ligands to carbonic anhydrase activatorsErica Vigiani, Alessandro Bonardi, Daniela Catarzi, et al.Pageof 29