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Journal of Enzyme Inhibition and Medicinal Chemistry|March 20, 2020
S-substituted 2-mercaptoquinazolin-4(3H)-one and 4-ethylbenzensulfonamides act as potent and selective human carbonic anhydrase IX and XII inhibitorsAdel S El-Azab, Alaa A-M Abdel-Aziz, Silvia Bua, et al.
Molecules (Basel, Switzerland)|November 26, 2022
Carbonic Anhydrase Inhibition Activities of Schiff's Bases Based on Quinazoline-Linked BenzenesulfonamideAdel S El-Azab, Alaa A-M Abdel-Aziz, Hazem A Ghabbour, et al.
European Journal of Medicinal Chemistry|December 17, 2021
2-(2-Hydroxyethyl)piperazine derivatives as potent human carbonic anhydrase inhibitors: Synthesis, enzyme inhibition, computational studies and antiglaucoma activityNiccolò Chiaramonte, Andrea Angeli, Silvia Sgambellone, et al.
Journal of Enzyme Inhibition and Medicinal Chemistry|March 21, 2022
The three-tails approach as a new strategy to improve selectivity of action of sulphonamide inhibitors against tumour-associated carbonic anhydrase IX and XIIAlessandro Bonardi, Silvia Bua, Jacob Combs, et al.
European Journal of Medicinal Chemistry|November 14, 2019
Synthesis, biological and molecular dynamics investigations with a series of triazolopyrimidine/triazole-based benzenesulfonamides as novel carbonic anhydrase inhibitorsMohamed A Said, Wagdy M Eldehna, Alessio Nocentini, et al.
European Journal of Medicinal Chemistry|May 13, 2022
Development of 4-((3-oxo-3-phenylpropyl)amino)benzenesulfonamide derivatives utilizing tail/dual-tail approaches as novel carbonic anhydrase inhibitorsMostafa M Elbadawi, Wagdy M Eldehna, Alessio Nocentini, et al.
International Journal of Biological Macromolecules|August 13, 2025
2-(Piperidin-1-yl)-N-(4-sulfamoylphenyl)acetamide derivatives as novel inhibitors of cancer-associated carbonic anhydrase isoforms IX and XIIWagdy M Eldehna, Mostafa M Elbadawi, Zainab M Elsayed, et al.
Journal of Medicinal Chemistry|May 22, 2024
Development of Penicillin-Based Carbonic Anhydrase Inhibitors Targeting Multidrug-Resistant Neisseria gonorrhoeaeAlessandro Bonardi, Alessio Nocentini, Simone Giovannuzzi, et al.
Journal of Medicinal Chemistry|December 3, 2025
Identification of Benzenesulfonamide-Containing Thiazolidine-2,4-Dione Derivatives as Novel Carbonic Anhydrase II and VII Inhibitors with Anti-Epileptic ActivityMohamed M Eldesouki, Mahmoud Abdelrahman Alkabbani, Mohammed S Taghour, et al.
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