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Journal of Enzyme Inhibition and Medicinal Chemistry|November 10, 2025
Harnessing coumarin-thio(seleno)cyanate conjugates: potent In vivo antiproliferative agents targeting carbonic anhydrasesSilvia Alejandra Meza-Ireta, Laura L Romero-Hernández, Paloma Begines, et al.ACS Infectious Diseases|March 25, 2021
Structure-Activity Relationship Studies of Acetazolamide-Based Carbonic Anhydrase Inhibitors with Activity against Neisseria gonorrhoeaeChad S Hewitt, Nader S Abutaleb, Ahmed E M Elhassanny, et al.Journal of Medicinal Chemistry|May 6, 2026
Structure-Activity Relationship Studies for 1,3,4-Thiadiazole-Based Bacterial Carbonic Anhydrase Inhibitors with In Vivo Efficacy against Drug-Resistant Neisseria gonorrhoeaePrabhakara R Tharra, Molly S Youse, Nader S Abutaleb, et al.International Journal of Biological Macromolecules|February 22, 2026
Trypanosoma cruzi carbonic anhydrase inhibitors as a potential antiparasitic agentSarah da Costa Lanera, Leonardo da Silva Lara, Lorraine Martins Rocha Orlando, et al.Journal of Medicinal Chemistry|October 30, 2023
4-(3-Phenyl-4-(3,4,5-trimethoxybenzoyl)-1H-pyrrol-1-yl)benzenesulfonamide, a Novel Carbonic Anhydrase and Wnt/β-Catenin Signaling Pathway Dual-Targeting Inhibitor with Potent Activity against Multidrug Resistant Cancer CellsDomiziana Masci, Michela Puxeddu, Laura Di Magno, et al.ACS Infectious Diseases|December 11, 2025
Bacterial Carbonic Anhydrase Inhibitor CAI0019 Demonstrates Efficacy in Enterococcus faecium Septicemic Peritonitis Mouse Model While Sparing the MicrobiomeNader S Abutaleb, Katrina J Holly, Carolyn K Metcalfe, et al.Pageof 29