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Journal of Enzyme Inhibition and Medicinal Chemistry|September 18, 2018
Steroids interfere with human carbonic anhydrase activity by using alternative binding mechanismsAlessio Nocentini, Alessandro Bonardi, Paola Gratteri, et al.
Magnetic Resonance in Chemistry : MRC|March 23, 2026
Quantitative Competition Binding of Fluorinated Ligands by Real-Time 19F In-Cell NMR to Assess Isoform Selectivity in Human CellsAzzurra Costantino, Letizia Barbieri, Simone Giovannuzzi, et al.
Journal of Enzyme Inhibition and Medicinal Chemistry|May 18, 2021
Biochemical profiling of anti-HIV prodrug Elsulfavirine (Elpida®) and its active form VM1500A against a panel of twelve human carbonic anhydrase isoformsClaudiu T Supuran, Alessio Nocentini, Elena Yakubova, et al.
ACS Medicinal Chemistry Letters|January 15, 2025
Tetrazole Is a Novel Zinc Binder Chemotype for Carbonic Anhydrase InhibitionSimone Giovannuzzi, Andrea Angeli, Paloma Begines, et al.
Journal of Enzyme Inhibition and Medicinal Chemistry|September 1, 2023
Aryl derivatives of 3H-1,2-benzoxaphosphepine 2-oxides as inhibitors of cancer-related carbonic anhydrase isoforms IX and XIIAnastasija Balašova, Aleksandrs Pustenko, Alessio Nocentini, et al.
Bioorganic & Medicinal Chemistry|January 27, 2019
α-Carbonic anhydrases are strongly activated by spinaceamine derivativesSuleyman Akocak, Nabih Lolak, Silvia Bua, et al.
Angewandte Chemie (International Ed. in English)|February 6, 2020
Drug Screening in Human Cells by NMR Spectroscopy Allows the Early Assessment of Drug PotencyEnrico Luchinat, Letizia Barbieri, Matteo Cremonini, et al.
ACS Chemical Biology|September 21, 2020
Intracellular Binding/Unbinding Kinetics of Approved Drugs to Carbonic Anhydrase II Observed by in-Cell NMREnrico Luchinat, Letizia Barbieri, Matteo Cremonini, et al.
Journal of Enzyme Inhibition and Medicinal Chemistry|January 6, 2022
Pharmaceutical strategies for preventing toxicity and promoting antioxidant and anti-inflammatory actions of bilirubinAlessio Nocentini, Alessandro Bonardi, Simone Pratesi, et al.
European Journal of Medicinal Chemistry|September 1, 2019
Structure-activity relationship with pyrazoline-based aromatic sulfamates as carbonic anhydrase isoforms I, II, IX and XII inhibitors: Synthesis and biological evaluationDavide Moi, Alessio Nocentini, Alessandro Deplano, et al.
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