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Journal of Medicinal Chemistry|December 5, 2017
Discovery and Optimization of Thiazolidinyl and Pyrrolidinyl Derivatives as Inhaled PDE4 Inhibitors for Respiratory DiseasesLaura Carzaniga, Gabriele Amari, Andrea Rizzi, et al.Journal of Biomedical Science|February 19, 2025
K27-linked RORγt ubiquitination by Nedd4 potentiates Th17-mediated autoimmunityQiuming Zeng, Hui Guo, Na Tang, et al.International Journal of Cancer|June 6, 2025
Combination therapy with levofloxacin and the probiotic Clostridium butyricum MIYAIRI 588 enhances immune checkpoint inhibitor efficacyKohei Tajima, Masahiro Hosonuma, Eiji Funayama, et al.Microbiology Spectrum|January 16, 2025
Association between the <i>ABCC11</i> gene polymorphism-determined earwax properties and external auditory canal microbiota in healthy adultsYasunobu Amari, Masahiro Hosonuma, Takuya Mizukami, et al.Journal of Medicinal Chemistry|August 10, 2023
Optimization of M<sub>3</sub> Antagonist-PDE4 Inhibitor (MAPI) Dual Pharmacology Molecules for the Treatment of COPDAndrea Rizzi, Gabriele Amari, Fausto Pivetti, et al.Nature Communications|June 1, 2023
Increased renal elimination of endogenous and synthetic pyrimidine nucleosides in concentrative nucleoside transporter 1 deficient miceAvinash K Persaud, Matthew C Bernier, Michael A Massey, et al.Cell Death Discovery|April 13, 2025
An in vivo "turning model" reveals new RanBP9 interactions in lung macrophagesYasuko Kajimura, Shuxin Dong, Anna Tessari, et al.Journal of Medicinal Chemistry|June 18, 2021
Discovery of M<sub>3</sub> Antagonist-PDE4 Inhibitor Dual Pharmacology Molecules for the Treatment of Chronic Obstructive Pulmonary DiseaseElisabetta Armani, Andrea Rizzi, Carmelida Capaldi, et al.Journal of Medicinal Chemistry|January 10, 2014
Novel class of benzoic acid ester derivatives as potent PDE4 inhibitors for inhaled administration in the treatment of respiratory diseasesElisabetta Armani, Gabriele Amari, Andrea Rizzi, et al.Biorxiv : the Preprint Server for Biology|February 24, 2023
Oncogenic Kras <sup>G12D</sup> specific non-covalent inhibitor reprograms tumor microenvironment to prevent and reverse early pre-neoplastic pancreatic lesions and in combination with immunotherapy regresses advanced PDAC in a CD8 <sup>+</sup> T cells dependent mannerKrishnan K Mahadevan, Kathleen M McAndrews, Valerie S LeBleu, et al.Pageof 91