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Journal of Medicinal Chemistry|August 26, 2021
Discovery and Structure-Activity Relationships of Quinazolinone-2-carboxamide Derivatives as Novel Orally Efficacious AntimalarialsBenoît Laleu, Yuichiro Akao, Atsuko Ochida, et al.Journal of Medicinal Chemistry|October 31, 2018
Target Validation and Identification of Novel Boronate Inhibitors of the Plasmodium falciparum ProteasomeStanley C Xie, David L Gillett, Natalie J Spillman, et al.Journal of Medicinal Chemistry|January 23, 2014
2,4-Diaminothienopyrimidines as orally active antimalarial agentsDiego González Cabrera, Claire Le Manach, Frederic Douelle, et al.Antimicrobial Agents and Chemotherapy|November 26, 2014
Histone methyltransferase inhibitors are orally bioavailable, fast-acting molecules with activity against different species causing malaria in humansNicholas A Malmquist, Sandeep Sundriyal, Joachim Caron, et al.Journal of Medicinal Chemistry|March 24, 2021
Discovery of Potent and Fast-Acting Antimalarial Bis-1,2,4-triazinesDaniel L Priebbenow, Mitch Mathiew, Da-Hua Shi, et al.Mbio|May 8, 2024
On-target, dual aminopeptidase inhibition provides cross-species antimalarial activityRebecca C S Edgar, Tess R Malcolm, Ghizal Siddiqui, et al.Nature Microbiology|August 16, 2017
Hexahydroquinolines are antimalarial candidates with potent blood-stage and transmission-blocking activityManu Vanaerschot, Leonardo Lucantoni, Tao Li, et al.Journal of Medicinal Chemistry|September 16, 2016
Discovery of a Quinoline-4-carboxamide Derivative with a Novel Mechanism of Action, Multistage Antimalarial Activity, and Potent in Vivo EfficacyBeatriz Baragaña, Neil R Norcross, Caroline Wilson, et al.Chemmedchem|June 13, 2019
Substituted Aminoacetamides as Novel Leads for Malaria TreatmentNeil R Norcross, Caroline Wilson, Beatriz Baragaña, et al.ACS Infectious Diseases|April 30, 2021
Repositioning and Characterization of 1-(Pyridin-4-yl)pyrrolidin-2-one Derivatives as Plasmodium Cytoplasmic Prolyl-tRNA Synthetase InhibitorsMasanori Okaniwa, Akira Shibata, Atsuko Ochida, et al.Pageof 22