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Chemmedchem|February 4, 2026
Structure-Based Discovery of Obeticholic Acid Derivatives as Novel Farnesoid X Receptor Partial Agonists with Improved Selectivity and Reduced Off-Target EffectsDaniela Passeri, Bruno Cerra, Andrea Carotti, et al.Bioorganic & Medicinal Chemistry|May 9, 2012
Pyrazole[3,4-e][1,4]thiazepin-7-one derivatives as a novel class of Farnesoid X Receptor (FXR) agonistsMaura Marinozzi, Andrea Carotti, Emanuele Sansone, et al.European Journal of Medicinal Chemistry|October 10, 2014
Scaffold hopping approach on the route to selective tankyrase inhibitorsParide Liscio, Andrea Carotti, Stefania Asciutti, et al.Journal of Medicinal Chemistry|October 10, 2013
Synthesis and biological evaluation of direct thrombin inhibitors bearing 4-(piperidin-1-yl)pyridine at the P1 position with potent anticoagulant activityModesto de Candia, Filomena Fiorella, Gianfranco Lopopolo, et al.International Journal of Molecular Sciences|April 12, 2022
Critical Assessment of a Structure-Based Screening Campaign for IDO1 Inhibitors: Tips and PitfallsAndrea Mammoli, Elisa Bianconi, Luana Ruta, et al.Journal of Medicinal Chemistry|September 23, 2016
Discovery of 3α,7α,11β-Trihydroxy-6α-ethyl-5β-cholan-24-oic Acid (TC-100), a Novel Bile Acid as Potent and Highly Selective FXR Agonist for Enterohepatic DisordersRoberto Pellicciari, Daniela Passeri, Francesca De Franco, et al.Bioorganic & Medicinal Chemistry|August 17, 2024
Novel multitarget directed ligands inspired by riluzole: A serendipitous synthesis of substituted benzo[b][1,4]thiazepines potentially useful as neuroprotective agentsSamuele Maramai, Mario Saletti, Marco Paolino, et al.European Journal of Medicinal Chemistry|August 6, 2022
Novel analgesic/anti-inflammatory agents: 1,5-Diarylpyrrole nitrooxyethyl sulfides and related compounds as Cyclooxygenase-2 inhibitors containing a nitric oxide donor moiety endowed with vasorelaxant propertiesMario Saletti, Samuele Maramai, Annalisa Reale, et al.Pageof 10