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ACS Omega|July 17, 2023
Exploring the 5-Substituted 2-Aminobenzothiazole-Based DNA Gyrase B Inhibitors Active against ESKAPE PathogensMaša Sterle, Martina Durcik, Clare E M Stevenson, et al.RSC Advances|September 9, 2024
New N-phenylpyrrolamide inhibitors of DNA gyrase with improved antibacterial activityAndrej Emanuel Cotman, Federica Fulgheri, Martina Piga, et al.European Journal of Medicinal Chemistry|July 25, 2024
Development of narrow-spectrum topoisomerase-targeting antibacterials against mycobacteriaMaša Sterle, Eva Habjan, Martina Piga, et al.European Journal of Medicinal Chemistry|September 5, 2024
Improved N-phenylpyrrolamide inhibitors of DNA gyrase as antibacterial agents for high-priority bacterial strainsNace Zidar, Alessia Onali, Peter Peršolja, et al.Bioorganic & Medicinal Chemistry|June 21, 2024
Exploring the interaction of N-(benzothiazol-2-yl)pyrrolamide DNA gyrase inhibitors with the GyrB ATP-binding site lipophilic floor: A medicinal chemistry and QTAIM studyNace Zidar, Andrej Emanuel Cotman, Wessel Sinnige, et al.Biomedicine & Pharmacotherapy = Biomedecine & Pharmacotherapie|January 15, 2026
New mitochondrial KV1.3 conjugates are potent and specific inducers of apoptosis in cancer modelsŠpela Gubič, Marzia Fois, Xiaoyi Shi, et al.Angewandte Chemie (International Ed. in English)|May 20, 2026
Mitochondria-Targeting Moieties Based on N-Tethered Pyridinium CationsIvan Džajić, Natalija Trunkelj, Jernej Repas, et al.Journal of Medicinal Chemistry|January 12, 2023
Discovery and Hit-to-Lead Optimization of Benzothiazole Scaffold-Based DNA Gyrase Inhibitors with Potent Activity against Acinetobacter baumannii and Pseudomonas aeruginosaAndrej Emanuel Cotman, Martina Durcik, Davide Benedetto Tiz, et al.Journal of Medicinal Chemistry|March 6, 2023
New Dual Inhibitors of Bacterial Topoisomerases with Broad-Spectrum Antibacterial Activity and In Vivo Efficacy against Vancomycin-Intermediate Staphylococcus aureusMartina Durcik, Andrej Emanuel Cotman, Žan Toplak, et al.Pageof 3