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Future Medicinal Chemistry|December 9, 2020
The promise and current status of CDK12/13 inhibition for the treatment of cancerSolomon Tadesse, Derek R Duckett, Andrii Monastyrskyi
The Journal of Organic Chemistry|January 7, 2015
Metal-free arylation of ethyl acetoacetate with hypervalent diaryliodonium salts: an immediate access to diverse 3-aryl-4(1H)-quinolonesAndrii Monastyrskyi, Niranjan K Namelikonda, Roman Manetsch
Current Topics in Medicinal Chemistry|August 14, 2014
4(1H)-pyridone and 4(1H)-quinolone derivatives as antimalarials with erythrocytic, exoerythrocytic, and transmission blocking activitiesAndrii Monastyrskyi, Dennis E Kyle, Roman Manetsch
Biophysical Journal|May 19, 2024
Structure-independent machine-learning predictions of the CDK12 interactomeAleksandra Karolak, Konstancja Urbaniak, Andrii Monastyrskyi, et al.
Bioorganic & Medicinal Chemistry Letters|December 27, 2017
Discovery of 2-arylquinazoline derivatives as a new class of ASK1 inhibitorsAndrii Monastyrskyi, Simon Bayle, Victor Quereda, et al.
Journal of Medicinal Chemistry|September 11, 2010
Endochin optimization: structure-activity and structure-property relationship studies of 3-substituted 2-methyl-4(1H)-quinolones with antimalarial activityR Matthew Cross, Andrii Monastyrskyi, Tina S Mutka, et al.
Bioorganic & Medicinal Chemistry|January 1, 2018
Development of dual casein kinase 1δ/1ε (CK1δ/ε) inhibitors for treatment of breast cancerAndrii Monastyrskyi, Napon Nilchan, Victor Quereda, et al.
Cancer Cell|November 1, 2019
Therapeutic Targeting of CDK12/CDK13 in Triple-Negative Breast CancerVictor Quereda, Simon Bayle, Francesca Vena, et al.
Cancer Research Communications|June 4, 2026
Targeting GSTZ1 sensitizes KRAS G12C-mutant lung cancer cells by overcoming glutathione and glycolysis pathway rewiringYi Liao, Xueli Li, Min Liu, et al.
The Journal of Biological Chemistry|November 28, 2023
The reversible inhibitor SR-4835 binds Cdk12/cyclin K in a noncanonical G-loop conformationMaximilian Schmitz, Ines H Kaltheuner, Kanchan Anand, et al.
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