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ACS Medicinal Chemistry Letters|August 25, 2017
<i>N</i>-Acylbenzenesulfonamide Dihydro-1,3,4-oxadiazole Hybrids: Seeking Selectivity toward Carbonic Anhydrase IsoformsGiulia Bianco, Rita Meleddu, Simona Distinto, et al.Antiviral Research|December 9, 2019
Discovery of dihydroxyindole-2-carboxylic acid derivatives as dual allosteric HIV-1 Integrase and Reverse Transcriptase associated Ribonuclease H inhibitorsFrancesca Esposito, Mario Sechi, Nicolino Pala, et al.European Journal of Medicinal Chemistry|April 12, 2023
Broad-spectrum coronavirus 3C-like protease peptidomimetic inhibitors effectively block SARS-CoV-2 replication in cells: Design, synthesis, biological evaluation, and X-ray structure determinationIrina Stefanelli, Angela Corona, Carmen Cerchia, et al.Journal of Medicinal Chemistry|January 29, 2015
Structure-activity relationship of pyrrolyl diketo acid derivatives as dual inhibitors of HIV-1 integrase and reverse transcriptase ribonuclease H domainGiuliana Cuzzucoli Crucitti, Mathieu Métifiot, Luca Pescatori, et al.Viruses|May 27, 2023
DHFR Inhibitors Display a Pleiotropic Anti-Viral Activity against SARS-CoV-2: Insights into the Mechanisms of ActionDaniela Iaconis, Francesca Caccuri, Candida Manelfi, et al.Chemmedchem|May 23, 2014
Design, synthesis, and biological evaluation of 1,3-diarylpropenones as dual inhibitors of HIV-1 reverse transcriptaseRita Meleddu, Valeria Cannas, Simona Distinto, et al.Antiviral Research|August 10, 2023
Diketo acid inhibitors of nsp13 of SARS-CoV-2 block viral replicationAngela Corona, Valentina Noemi Madia, Riccardo De Santis, et al.European Journal of Medicinal Chemistry|August 24, 2019
Chromenone derivatives as a versatile scaffold with dual mode of inhibition of HIV-1 reverse transcriptase-associated Ribonuclease H function and integrase activityFrancesca Esposito, Francesca Alessandra Ambrosio, Rita Maleddu, et al.Journal of Enzyme Inhibition and Medicinal Chemistry|August 12, 2025
<i>N</i>-alkyl and <i>N</i>-benzyl indoles are anti-SARS-CoV-2 agents and nsp13 inhibitorsAurora Albano, Roberta Emmolo, Riccardo De Santis, et al.ACS Medicinal Chemistry Letters|May 16, 2022
Discovery of 2-Phenylquinolines with Broad-Spectrum Anti-coronavirus ActivityMaria Giulia Nizi, Leentje Persoons, Angela Corona, et al.Pageof 12