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Chemmedchem|May 5, 2025
Structure-Activity Relationships of New 1-Aryl-1H-Indole Derivatives as SARS-CoV-2 Nsp13 InhibitorsValentina Noemi Madia, Roberta Emmolo, Elisa Patacchini, et al.Journal of Medicinal Chemistry|June 9, 2021
Quinolinonyl Non-Diketo Acid Derivatives as Inhibitors of HIV-1 Ribonuclease H and Polymerase Functions of Reverse TranscriptaseAntonella Messore, Angela Corona, Valentina Noemi Madia, et al.ACS Pharmacology & Translational Science|January 16, 2025
Thiol-Reactive or Redox-Active: Revising a Repurposing Screen Led to a New Invalidation Pipeline and Identified a True Noncovalent Inhibitor Against Papain-like Protease from SARS-CoV-2Maria Kuzikov, Stefano Morasso, Jeanette Reinshagen, et al.ACS Medicinal Chemistry Letters|May 22, 2020
Pyrrolyl Pyrazoles as Non-Diketo Acid Inhibitors of the HIV-1 Ribonuclease H Function of Reverse TranscriptaseAntonella Messore, Angela Corona, Valentina Noemi Madia, et al.Antiviral Research|February 20, 2025
The efficiency of high-throughput screening (HTS) and in-silico data analysis during medical emergencies: Identification of effective antiviral 3CLpro inhibitorsDebora Zian, Daniela Iaconis, Simone Nenci, et al.Journal of Medicinal Chemistry|April 2, 2014
Basic quinolinonyl diketo acid derivatives as inhibitors of HIV integrase and their activity against RNase H function of reverse transcriptaseRoberta Costi, Mathieu Métifiot, Suhman Chung, et al.Chemmedchem|April 10, 2026
2-Phenylquinolines Exhibit Anti-Severe Acute Respiratory Syndrome Coronavirus-2 Activity Through the Nonstructural Protein 13 Helicase InhibitionGiada Cernicchi, Maria Giulia Nizi, Roberta Emmolo, et al.ACS Infectious Diseases|August 3, 2024
4-(3-Phenylsulfonylindol-2-yl)-1-(pyridin-2-yl)piperazinyl-methanones as Potent Inhibitors of both SARS-CoV-2 and HCoV-OC43 VirusesMichela Puxeddu, Manuela Donalisio, Joachim Jakob Bugert, et al.Pharmaceuticals (Basel, Switzerland)|May 25, 2024
New Thiazolidine-4-One Derivatives as SARS-CoV-2 Main Protease InhibitorsAntonella Messore, Paolo Malune, Elisa Patacchini, et al.Scientific Data|July 13, 2022
Cytopathic SARS-CoV-2 screening on VERO-E6 cells in a large-scale repurposing effortAndrea Zaliani, Laura Vangeel, Jeanette Reinshagen, et al.Pageof 12